1. Silverman, R.B. Mechanism-Based Enzyme Inactivation: Chemistry and Enzymology, Vols. I and II; CRC Press: Boca Raton, FL; 1988.

2a. Silverman, R.B. The Organic Chemistry of Drug Design and Drug Action; Academic Press: San Diego; 1992.

2b. Silverman, R. B. Medizinische Chemie für Organiker, Biochemiker und Pharmazeutische Chemiker, VCH: Weinheim; 1995 (German Translation by Joachim K. Seydel of The Organic Chemistry of Drug Design and Drug Action).

3. Silverman, R. B. The Organic Chemistry of Enzyme-Catalyzed Reactions, Academic Press: San Diego; 2000; revised, 2002.

4. Silverman, R.B. The Organic Chemistry of Drug Design and Drug Action; 2nd Edition; Elsevier/Academic Press: San Diego; 2004.